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EPZ-6438

EPZ-6438

CAS No:1403254-99-8 Catalog No.:HY-13803

Brief Description:

Price and Availability: 10 mM * 1 mL €69 ( In-stock ); 5mg €55 ( In-stock ); 10mg €77 ( In-stock ); 50mg €164 ( In-stock ); 100mg €262 ( In-stock ); 200mg €481 ( In-stock );

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GSK126

GSK126

CAS No:1346574-57-9 Catalog No.:HY-13470

Brief Description:

Price and Availability: 10 mM * 1 mL €76 ( In-stock ); 5mg €66 ( In-stock ); 10mg €98 ( In-stock ); 50mg €262 ( In-stock ); 100mg €437 ( In-stock ); 200mg €722 ( In-stock );

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GSK343

GSK343

CAS No:1346704-33-3 Catalog No.:HY-13500

Brief Description:

Price and Availability: 10 mM * 1 mL €66 ( In-stock ); 5mg €55 ( In-stock ); 10mg €87 ( In-stock ); 25mg €180 ( In-stock ); 50mg €306 ( In-stock ); 100mg €536 ( In-stock );

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UNC0642

UNC0642

CAS No:1481677-78-4 Catalog No.:HY-13980

Brief Description:

Price and Availability: 10 mM * 1 mL €118 ( In-stock ); 5mg €98 ( In-stock ); 10mg €164 ( In-stock ); 50mg €492 ( In-stock ); 100mg €929 ( In-stock );

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3-Deazaneplanocin A hydrochloride

3-Deazaneplanocin A hydrochloride

CAS No:120964-45-6 Catalog No.:HY-12186

Brief Description:

Price and Availability: 10 mM * 1 mL €323 ( In-stock ); 1mg €98 ( In-stock ); 5mg €361 ( In-stock ); 10mg €547 ( In-stock ); 25mg €984 ( In-stock );

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UNC1999

UNC1999

CAS No:1431612-23-5 Catalog No.:HY-15646

Brief Description:

Price and Availability: 10 mM * 1 mL €94 ( In-stock ); 5mg €75 ( In-stock ); 10mg €131 ( In-stock ); 50mg €394 ( In-stock ); 100mg €700 ( In-stock );

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EPZ-5676

EPZ-5676

CAS No:1380288-87-8 Catalog No.:HY-15593

Brief Description:

Price and Availability: 10 mM * 1 mL €162 ( In-stock ); 5mg €131 ( In-stock ); 10mg €175 ( In-stock ); 50mg €634 ( In-stock );

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EPZ015666

EPZ015666

CAS No:1616391-65-1 Catalog No.:HY-12727

Brief Description:

Price and Availability: 10 mM * 1 mL €192 ( In-stock ); 5mg €175 ( In-stock ); 10mg €279 ( In-stock ); 50mg €1071 ( In-stock );

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EPZ004777

EPZ004777

CAS No:1338466-77-5 Catalog No.:HY-15227

Brief Description:

Price and Availability: 10 mM * 1 mL €143 ( In-stock ); 5mg €120 ( In-stock ); 10mg €208 ( In-stock ); 50mg €601 ( In-stock ); 100mg €1028 ( In-stock );

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BIX-01294

BIX-01294

CAS No:935693-62-2 Catalog No.:HY-10587

Brief Description:

Price and Availability: 10 mM * 1 mL €149 ( In-stock ); 10mg €136 ( In-stock ); 50mg €453 ( In-stock );

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EPZ031686

EPZ031686

CAS No:1808011-22-4 Catalog No.:HY-19324

Brief Description: EPZ031686 is a noncompetitive inhibitor for SMYD3 and MEKK2 with a Ki=1.2 and 1.1 nM respectively.

Price and Availability: 10 mM * 1 mL €497 ( In-stock ); 1mg €164 ( In-stock ); 5mg €383 ( In-stock ); 10mg €547 ( In-stock ); 50mg €1640 ( In-stock ); 100mg €2296 ( In-stock );

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UNC0638

UNC0638

CAS No:1255580-76-7 Catalog No.:HY-15273

Brief Description:

Price and Availability: 10 mM * 1 mL €74 ( In-stock ); 5mg €66 ( In-stock ); 10mg €98 ( In-stock ); 50mg €273 ( In-stock ); 100mg €481 ( In-stock );

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EPZ015866

EPZ015866

CAS No:1616391-87-7 Catalog No.:HY-100235

Brief Description: EPZ015866 (GSK591) is a potent selective inhibitor of the arginine methyltransferase PRMT5. It maintained excellent selectivity against other PMT enzymes observed with EPZ015666 [1].

Price and Availability: 10 mM * 1 mL €132 ( In-stock ); 5mg €120 ( In-stock ); 10mg €197 ( In-stock ); 25mg €404 ( In-stock ); 50mg €678 ( In-stock ); 100mg €1039 ( In-stock );

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LLY-507

LLY-507

CAS No:1793053-37-8 Catalog No.:HY-19313

Brief Description: LLY-507 is a potent inhibitor of SMYD2 with IC50 < 15 nM, is >100-fold selective for SMYD2 over a broad range of methyltransferase and non-methyltransferase targets.

Price and Availability: 10 mM * 1 mL €138 ( In-stock ); 5mg €109 ( In-stock ); 10mg €197 ( In-stock ); 25mg €426 ( In-stock ); 50mg €765 ( In-stock );

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A-366

A-366

CAS No:1527503-11-2 Catalog No.:HY-12583

Brief Description: A-366 is a peptide-competitive inhibitor of G9a/GLP with an enzymatic IC50 of ~3 nM and >100-fold selectivity over other methyltransferases and other non-epigenetic targets.

Price and Availability: 10 mM * 1 mL €78 ( In-stock ); 5mg €71 ( In-stock ); 10mg €120 ( In-stock ); 50mg €481 ( In-stock );

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MS023

MS023

CAS No:1831110-54-3 Catalog No.:HY-19615

Brief Description: MS023 is a potent, selective, and cell-active inhibitor of human type I PRMTs with IC50 of 4-119 nM.

Price and Availability: 10 mM * 1 mL €138 ( In-stock ); 2mg €87 ( In-stock ); 5mg €120 ( In-stock ); 10mg €197 ( In-stock ); 25mg €361 ( In-stock ); 50mg €667 ( In-stock ); 100mg €1203 ( In-stock );

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AZ505 ditrifluoroacetate

AZ505 ditrifluoroacetate

CAS No:1035227-44-1 Catalog No.:HY-15226A

Brief Description: AZ505 ditrifluoroacetate is a potent and highly selective inhibitor of the oncogenic protein SMYD2(IC50=0.12 uM) with potential anticancer activity, >600 fold than SMYD3(IC50>83.3 uM); DOT1L(IC50>83.3 uM);EZH2(IC50>83.3 uM).

Price and Availability: 10 mM * 1 mL €310 ( In-stock ); 5mg €208 ( In-stock ); 10mg €350 ( In-stock ); 25mg €743 ( In-stock ); 50mg €1082 ( In-stock ); 100mg €1640 ( In-stock );

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GSK3326595

GSK3326595

CAS No:1616392-22-3 Catalog No.:HY-101563

Brief Description:

Price and Availability: 10 mM * 1 mL €84 ( In-stock ); 5mg €77 ( In-stock ); 10mg €131 ( In-stock ); 50mg €383 ( In-stock ); 100mg €656 ( In-stock ); 200mg €1203 ( In-stock );

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SGC0946

SGC0946

CAS No:1561178-17-3 Catalog No.:HY-15650

Brief Description: SGC0946 is a highly potent and selective DOT1L methyltransferase inhibitor with IC50 of 0.3 nM; selectively kill mixed lineage leukaemia cells.

Price and Availability: 10 mM * 1 mL €89 ( In-stock ); 5mg €66 ( In-stock ); 10mg €115 ( In-stock ); 50mg €459 ( In-stock );

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GSK503

GSK503

CAS No:1346572-63-1 Catalog No.:HY-12856

Brief Description:

Price and Availability: 10 mM * 1 mL €114 ( In-stock ); 5mg €98 ( In-stock ); 10mg €142 ( In-stock ); 50mg €492 ( In-stock ); 100mg €875 ( In-stock );

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PFI-2 hydrochloride

PFI-2 hydrochloride

CAS No:1627607-87-7 Catalog No.:HY-18627A

Brief Description: PFI-2 hydrochloride is a a first-in-class, potent, highly selective, and cell-active inhibitor of the methyltransferase activity of SETD7 with IC50 of 2 nM, 500 fold active than (S)-PFI-2.

Price and Availability: 10 mM * 1 mL €169 ( In-stock ); 10mg €153 ( In-stock ); 50mg €492 ( In-stock );

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EPZ005687

EPZ005687

CAS No:1396772-26-1 Catalog No.:HY-15555

Brief Description:

Price and Availability: 10 mM * 1 mL €140 ( In-stock ); 5mg €118 ( In-stock ); 10mg €131 ( In-stock ); 50mg €306 ( In-stock ); 100mg €421 ( In-stock );

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EED226

EED226

CAS No:2083627-02-3 Catalog No.:HY-101117

Brief Description:

Price and Availability: 10 mM * 1 mL €144 ( In-stock ); 5mg €131 ( In-stock ); 10mg €208 ( In-stock ); 50mg €601 ( In-stock ); 100mg €1082 ( In-stock );

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UNC0321

UNC0321

CAS No:1238673-32-9 Catalog No.:HY-10930

Brief Description: UNC0321 is a potent and selective G9a inhibitor with Ki of 63 pM, UNC0321 is the first G9a inhibitor with picomolar potency and the most potent G9a inhibitor to date.

Price and Availability: 10 mM * 1 mL €120 ( In-stock ); 5mg €106 ( In-stock ); 10mg €164 ( In-stock ); 50mg €765 ( In-stock );

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OICR-9429

OICR-9429

CAS No:1801787-56-3 Catalog No.:HY-16993

Brief Description: OICR-9429 is a novel small-molecule antagonist of the Wdr5-MLL interaction with IC50 of 5 uM. inhibit proliferation and induce differentiation .

Price and Availability: 10 mM * 1 mL €107 ( In-stock ); 5mg €87 ( In-stock ); 10mg €131 ( In-stock ); 25mg €273 ( In-stock ); 50mg €492 ( In-stock ); 100mg €765 ( In-stock );

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EPZ020411 hydrochloride

EPZ020411 hydrochloride

CAS No: Catalog No.:HY-12970A

Brief Description: EPZ020411 hydrochloride is a potent and selective inhibitor of PRMT6 with IC50 of 10 nM, has >10 fold selectivity for PRMT6 over PRMT1 and PRMT8.

Price and Availability: 10 mM * 1 mL €184 ( In-stock ); 2mg €109 ( In-stock ); 5mg €175 ( In-stock ); 10mg €284 ( In-stock ); 50mg €1039 ( In-stock ); 100mg €1585 ( In-stock );

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AMI-1

AMI-1

CAS No:20324-87-2 Catalog No.:HY-18962

Brief Description: AMI-1 is a potent, cell-permeable compound which inhibits protein arginine N-methyltransferases (PRMTs), including human PRMT1 (IC50 = 8.8μM) and yeast-Hmt1p (IC50 = 3.0μM), by blocking peptide-substrate binding.

Price and Availability: 10 mM * 1 mL €99 ( In-stock ); 5mg €82 ( In-stock ); 10mg €131 ( In-stock ); 25mg €262 ( In-stock );

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MS049

MS049

CAS No:1502816-23-0 Catalog No.:HY-100360

Brief Description: MS 049 is a potent, selective, and cell-active dual inhibitor of PRMT4 and PRMT6 with IC 50 of 34 nM and 43 nM respectively.

Price and Availability: 10 mM * 1 mL €72 ( In-stock ); 5mg €66 ( In-stock ); 10mg €109 ( In-stock ); 25mg €241 ( In-stock ); 50mg €437 ( In-stock ); 100mg €820 ( In-stock );

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Chaetocin

Chaetocin

CAS No:28097-03-2 Catalog No.:HY-N2019

Brief Description:

Price and Availability: 10 mM * 1 mL €754 ( In-stock ); 1mg €164 ( In-stock ); 5mg €492 ( In-stock ); 10mg €885 ( In-stock );

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UNC3866

UNC3866

CAS No:1872382-47-2 Catalog No.:HY-100832

Brief Description:

Price and Availability: 10 mM * 1 mL €200 ( In-stock ); 5mg €131 ( In-stock ); 10mg €230 ( In-stock ); 25mg €448 ( In-stock ); 50mg €831 ( In-stock ); 100mg €1476 ( In-stock );

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Amodiaquin dihydrochloride dihydrate

Amodiaquin dihydrochloride dihydrate

CAS No:6398-98-7 Catalog No.:HY-B1322

Brief Description: Amodiaquine dihydrochloride dihydrate is a histamine N-methyltransferase inhibitor, used as an antimalarial and anti-inflammatory agent.

Price and Availability: 10 mM * 1 mL €60 ( In-stock ); 100mg €55 ( In-stock );

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MM-102 trifluoroacetate

MM-102 trifluoroacetate

CAS No: Catalog No.:HY-12220A

Brief Description: MM-102 trifluoroacetate is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is >200 times more potent than the ARA peptide.

Price and Availability: 10 mM * 1 mL €169 ( In-stock ); 2mg €55 ( In-stock ); 5mg €120 ( In-stock ); 10mg €197 ( In-stock ); 50mg €831 ( In-stock );

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UNC1215

UNC1215

CAS No:1415800-43-9 Catalog No.:HY-15649

Brief Description: UNC1215 is a potent and selective chemical probe for the methyllysine (Kme) reading function of L3MBTL3 with Kd value of 120 nM.

Price and Availability: 10 mM * 1 mL €102 ( In-stock ); 5mg €87 ( In-stock ); 10mg €153 ( In-stock ); 50mg €562 ( In-stock );

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EI1

EI1

CAS No:1418308-27-6 Catalog No.:HY-15573

Brief Description:

Price and Availability: 10 mM * 1 mL €120 ( In-stock ); 5mg €109 ( In-stock ); 10mg €186 ( In-stock ); 50mg €568 ( In-stock ); 100mg €787 ( In-stock );

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UNC0646

UNC0646

CAS No:1320288-17-2 Catalog No.:HY-13807

Brief Description: UNC0646 is a potent and selective G9a inhibitor with IC50 of 6 nM.

Price and Availability: 10 mM * 1 mL €90 ( In-stock ); 5mg €66 ( In-stock ); 10mg €115 ( In-stock ); 50mg €384 ( In-stock );

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SGC707

SGC707

CAS No:1687736-54-4 Catalog No.:HY-19715

Brief Description: SGC707 is a first-in-class PRMT3 chemical probe which is a potent, selective, and cell-active allosteric inhibitor of PRMT3 with IC50 of 31 nM.

Price and Availability: 10 mM * 1 mL €72 ( In-stock ); 5mg €66 ( In-stock ); 10mg €98 ( In-stock ); 50mg €383 ( In-stock ); 100mg €656 ( In-stock );

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BCI-121

BCI-121

CAS No:432529-82-3 Catalog No.:HY-21972

Brief Description:

Price and Availability: 10 mM * 1 mL €72 ( In-stock ); 5mg €66 ( In-stock ); 10mg €104 ( In-stock ); 25mg €213 ( In-stock ); 50mg €372 ( In-stock ); 100mg €645 ( In-stock );

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UNC 0631

UNC 0631

CAS No:1320288-19-4 Catalog No.:HY-13808

Brief Description:

Price and Availability: 5mg €126 ( In-stock ); 10mg €219 ( In-stock ); 25mg €468 ( In-stock ); 50mg €742 ( In-stock );

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UNC0379

UNC0379

CAS No:1620401-82-2 Catalog No.:HY-12335

Brief Description: UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8 with IC50 of 7.3±1.0 uM; selective over 15 other methyltransferases.

Price and Availability: 10 mM * 1 mL €120 ( In-stock ); 5mg €109 ( In-stock ); 10mg €148 ( In-stock ); 50mg €443 ( In-stock ); 100mg €640 ( In-stock );

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CARM1-IN-1

CARM1-IN-1

CAS No:1020399-49-8 Catalog No.:HY-12759

Brief Description: CARM1-IN-1 is a potent and specific CARM1(Coactivator-associated arginine methyltransferase 1) inhibitor with IC50 of 8.6 uM; shows very low activity against PRMT1 and SET7(IC50 > 600 uM).

Price and Availability: 10 mM * 1 mL €467 ( In-stock ); 5mg €383 ( In-stock ); 10mg €711 ( In-stock ); 50mg €2186 ( In-stock );

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MI-2

MI-2

CAS No:1271738-62-5 Catalog No.:HY-15222

Brief Description: MI-2 is a Menin-MLL interaction inhibitor with IC50 value of 446 ± 28 nM.

Price and Availability: 10 mM * 1 mL €157 ( In-stock ); 5mg €142 ( In-stock ); 10mg €197 ( In-stock ); 50mg €547 ( In-stock ); 100mg €875 ( In-stock ); 200mg €1367 ( In-stock );

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EPZ011989

EPZ011989

CAS No:1598383-40-4 Catalog No.:HY-16986

Brief Description: EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.

Price and Availability: 10 mM * 1 mL €117 ( In-stock ); 5mg €87 ( In-stock ); 10mg €153 ( In-stock ); 50mg €372 ( In-stock ); 100mg €547 ( In-stock );

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UNC0224

UNC0224

CAS No:1197196-48-7 Catalog No.:HY-10929

Brief Description: UNC0224 is a potent and selective G9a inhibitor with IC50 of 15 nM in in the G9a Thioglo assay.

Price and Availability: 10 mM * 1 mL €117 ( In-stock ); 5mg €106 ( In-stock ); 10mg €164 ( In-stock ); 50mg €765 ( In-stock );

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MI-538

MI-538

CAS No:1857417-10-7 Catalog No.:HY-19810

Brief Description:

Price and Availability: 10 mM * 1 mL €327 ( In-stock ); 1mg €120 ( In-stock ); 5mg €262 ( In-stock ); 10mg €459 ( In-stock ); 25mg €918 ( In-stock ); 50mg €1257 ( In-stock ); 100mg €2132 ( In-stock );

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SGC2085

SGC2085

CAS No:1821908-48-8 Catalog No.:HY-100565

Brief Description:

Price and Availability: 10 mM * 1 mL €248 ( In-stock ); 1mg €120 ( In-stock ); 5mg €361 ( In-stock ); 10mg €547 ( In-stock ); 50mg €1640 ( In-stock ); 100mg €2296 ( In-stock );

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CPI-1205

CPI-1205

CAS No:1621862-70-1 Catalog No.:HY-100021

Brief Description:

Price and Availability: 10 mM * 1 mL €200 ( In-stock ); 2mg €98 ( In-stock ); 5mg €175 ( In-stock ); 10mg €306 ( In-stock ); 25mg €645 ( In-stock ); 50mg €1049 ( In-stock );

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MI-463

MI-463

CAS No:1628317-18-9 Catalog No.:HY-19809

Brief Description:

Price and Availability: 10 mM * 1 mL €175 ( In-stock ); 1mg €77 ( In-stock ); 5mg €164 ( In-stock ); 10mg €230 ( In-stock ); 50mg €514 ( In-stock ); 100mg €732 ( In-stock );

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C-7280948

C-7280948

CAS No:587850-67-7 Catalog No.:HY-15890

Brief Description: C-7280948 is a PRMT1 inhibitor.

Price and Availability: 10 mM * 1 mL €84 ( In-stock ); 10mg €77 ( In-stock ); 50mg €230 ( In-stock );

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WDR5-0103

WDR5-0103

CAS No:890190-22-4 Catalog No.:HY-19347

Brief Description: WDR5-0103 is a potent and selective WD repeat-containing protein 5 (WDR5) antagonist with Kd of 450 nM.

Price and Availability: 10 mM * 1 mL €72 ( In-stock ); 5mg €66 ( In-stock ); 10mg €109 ( In-stock ); 50mg €437 ( In-stock ); 100mg €711 ( In-stock );

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BRD9539

BRD9539

CAS No:1374601-41-8 Catalog No.:HY-15647

Brief Description: BRD9539 inhibits G9a activity with an IC50 of 6.3 μM, inhibits PRC2 activity with a similar IC50.

Price and Availability: 10 mM * 1 mL €84 ( In-stock ); 5mg €77 ( In-stock ); 10mg €131 ( In-stock ); 25mg €284 ( In-stock ); 50mg €503 ( In-stock );

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